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2004, Vol. 76, Issue 5

Polish-Austrian-German-Hungarian-Italian Joint Meeting on Medicinal Chemistry, Kraków, Poland, 15–18 October 2003

Predicting drug metabolism: Concepts and challenges
B. Testa, A.-L. Balmat and Anthony Long
p. 907 [Details + Abstract] [Full text - pdf 202 kB]
Prion protein as a target for therapeutic interventions
P. P. Liberski
p. 915 [Details + Abstract] [Full text - pdf 175 kB]
Structural basis for 2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid (AMPA) receptor activation
T. N. Johansen, J. R. Greenwood, S. B. Vogensen and Povl Krogsgaard-Larsen
p. 921 [Details + Abstract] [Full text - pdf 455 kB]
Search for noncompetitive 2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid receptor (AMPAR) antagonists: Synthesis, pharmacological properties, and computational studies
A. Chimirri, G. De Sarro, S. Quartarone, M. L. Barreca, R. Caruso, L. De Luca and R. Gitto
p. 931 [Details + Abstract] [Full text - pdf 381 kB]
Neuropeptide mimetics for pain management
A. W. Lipkowski, A. Misicka, D. B. Carr, G. Ronsisvalle, Dariusz Kosson and I. Maszczynska Bonney
p. 941 [Details + Abstract] [Full text - pdf 280 kB]
New endomorphin analogs with mu-agonist and delta-antagonist properties
G. Tóth, A. Keresztes, Cs. Tömböly, A. Péter, F. Fülöp, D. Tourwé, E. Navratilova, É. Varga, W. R. Roeske, H. I. Yamamura, M. Szucs and A. Borsodi
p. 951 [Details + Abstract] [Full text - pdf 208 kB]
Spacer conformation in biologically active molecules
J. Karolak-Wojciechowska and A. Fruzinski
p. 959 [Details + Abstract] [Full text - pdf 243 kB]
Discovery of new anti-inflammatory agents
F. Fülöp, László Lázár, Z. Szakonyi, M. Pihlavisto, Sakari Alaranta, P. J. Vainio, Auni Juhakoski, Anne Marjamäki and D. J. Smith
p. 965 [Details + Abstract] [Full text - pdf 238 kB]
NO donors: Focus on furoxan derivatives
A. Gasco, R. Fruttero, G. Sorba, A. Di Stilo and R. Calvino
p. 973 [Details + Abstract] [Full text - pdf 245 kB]
Passive and catalytic antibodies and drug delivery
G. M. Blackburn, J. H. Rickard, S. Cesaro-Tadic, D. Lagos, A. Mekhalfia, L. Partridge and A. Plückthun
p. 983 [Details + Abstract] [Full text - pdf 254 kB]
Virtual combinatorial chemistry and in silico screening: Efficient tools for lead structure discovery?
Thierry Langer and G. Wolber
p. 991 [Details + Abstract] [Full text - pdf 147 kB]
Development of modulators of multidrug resistance: A pharmacoinformatic approach
G. F. Ecker and Peter Chiba
p. 997 [Details + Abstract] [Full text - pdf 268 kB]
Hindered nucleoside analogs as antiflaviviridae agents
Stefano Manfredini, Angela Angusti, A. C. Veronese, Elisa Durini, S. Vertuani, F. Nalin, N. Solaroli, S. Pricl, Marco Ferrone, M. Mura, M. A. Piano, B. Poddesu, Alessandra Cadeddu, P. La Colla and Roberta Loddo
p. 1007 [Details + Abstract] [Full text - pdf 296 kB]
Solid- and solution-phase synthesis of bioactive dihydropyrimidines
D. Dallinger, A. Stadler and C. O. Kappe
p. 1017 [Details + Abstract] [Full text - pdf 244 kB]
Synthesis of naturally occurring o-heterocyclic compounds of biological activity
Sándor Antus, Katalin Gulácsi, László Juhász, Loránd Kiss and Tibor Kurtán
p. 1025 [Details + Abstract] [Full text - pdf 298 kB]

IUPAC Technical Reports and Recommendations

Glossary of terms used in toxicokinetics (IUPAC Recommendations 2003)
M. Nordberg, J. Duffus and D. M. Templeton
p. 1033 [Details + Abstract] [Full text - pdf 318 kB]