Pure and Applied Chemistry

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• LaPlante Steven R., Bös Michael, Brochu Christian, Chabot Catherine, Coulombe René, Gillard James R., Jakalian Araz, Poirier Martin, Rancourt Jean, Stammers Timothy, Thavonekham Bounkham, Beaulieu Pierre L., Kukolj George, Tsantrizos Youla S.: Conformation-Based Restrictions and Scaffold Replacements in the Design of Hepatitis C Virus Polymerase Inhibitors: Discovery of Deleobuvir (BI 207127). J. Med. Chem. 2014, 57, 1845. <http://dx.doi.org/10.1021/jm4011862>
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• Mykhailiuk Pavel K., Starova Viktoriia, Iurchenko Vladimir, Shishkina Svitlana V., Shishkin Oleg V., Khilchevskyi Oleksandr, Zaporozhets Olga: 1-Amino-4,4-difluorocyclohexanecarboxylic acid as a promising building block for drug discovery: design, synthesis and characterization. Tetrahedron 2013, 69, 4066. <http://dx.doi.org/10.1016/j.tet.2013.03.072>
• Okamoto Toru, Zobel Kerry, Fedorova Anna, Quan Clifford, Yang Hong, Fairbrother Wayne J., Huang David C. S., Smith Brian J., Deshayes Kurt, Czabotar Peter E.: Stabilizing the Pro-Apoptotic BimBH3 Helix (BimSAHB) Does Not Necessarily Enhance Affinity or Biological Activity. ACS Chem. Biol. 2013, 8, 297. <http://dx.doi.org/10.1021/cb3005403>
• Wang Yansong, Kirschner Alexander, Fabian Anne-Katrin, Gopalakrishnan Ranganath, Kress Christoph, Hoogeland Bastiaan, Koch Uwe, Kozany Christian, Bracher Andreas, Hausch Felix: Increasing the Efficiency of Ligands for FK506-Binding Protein 51 by Conformational Control. J. Med. Chem. 2013, 56, 3922. <http://dx.doi.org/10.1021/jm400087k>
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• Shi Yue, Zhu Crystal Z., Martin Stephen F., Ren Pengyu: Probing the Effect of Conformational Constraint on Phosphorylated Ligand Binding to an SH2 Domain Using Polarizable Force Field Simulations. Chem B 2012, 116, 1716. <http://dx.doi.org/10.1021/jp210265d>
• Aubé Jeffrey: Small-molecule libraries: Naturally inspired oligomers. Nature Chem 2012, 4, 71. <http://dx.doi.org/10.1038/nchem.1254>
• Lemmon Gordon, Kaufmann Kristian, Meiler Jens: Prediction of HIV-1 Protease/Inhibitor Affinity using RosettaLigand : HIV-1 Protease/Inhibitor Affinity Prediction. Chemical Biology and Drug Design 2012, 79, 888. <http://dx.doi.org/10.1111/j.1747-0285.2012.01356.x>
• Grygorenko Oleksandr O., Radchenko Dmytro S., Volochnyuk Dmitriy M., Tolmachev Andrey A., Komarov Igor V.: Bicyclic Conformationally Restricted Diamines. Chem. Rev. 2011, 111, 5506. <http://dx.doi.org/10.1021/cr100352k>
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• LaPlante Steven R., Gillard James R., Jakalian Araz, Aubry Norman, Coulombe René, Brochu Christian, Tsantrizos Youla S., Poirier Martin, Kukolj George, Beaulieu Pierre L.: Importance of Ligand Bioactive Conformation in the Discovery of Potent Indole-Diamide Inhibitors of the Hepatitis C Virus NS5B. J Am Chem Soc 2010, 132, 15204. <http://dx.doi.org/10.1021/ja101358s>
• Lee Yun-Young, Cho Sue-Kyung, Huh Jeong-Eun, Park Euddeum, Lee Soo-Young, Kwon Yong-Uk: Efficient Solid-Phase Synthesis of Peptoid Analogs for the Development of RANK Receptor Inhibitors. Bulletin of the Korean Chemical Society 2010, 31, 3437. <http://dx.doi.org/10.5012/bkcs.2010.31.11.3437>
• Sander Kerstin, Kottke Tim, Tanrikulu Yusuf, Proschak Ewgenij, Weizel Lilia, Schneider Erich H., Seifert Roland, Schneider Gisbert, Stark Holger: 2,4-Diaminopyrimidines as histamine H4 receptor ligands—Scaffold optimization and pharmacological characterization. biorg med chem 2009, 17, 7186. <http://dx.doi.org/10.1016/j.bmc.2009.08.059>
• Kwon Yong-Uk, Kodadek Thomas: Encoded combinatorial libraries for the construction of cyclic peptoid microarrays. Chem Commun 2008, 5704. <http://dx.doi.org/10.1039/b812735b>