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Pure Appl. Chem., 2001, Vol. 73, No. 9, pp. 1411-1420

http://dx.doi.org/10.1351/pac200173091411

New developments in A1 and A2 adenosine receptor antagonists

K. Kieć-Kononowicz1, A. Drabczyńska1, E. Pękala1, B. Michalak1, C. E. Müller2, B. Schumacher2, J. Karolak-Wojciechowska3, H. Duddeck4, S. Rockitt4 and R. Wartchow4

1 Jagiellonian University, Medical College, Department of Chemical Technology of Drugs, Medyczna 9, Pl 30-688 Kraków, Poland
2 Pharmaceutical Institute Poppelsdorf, University of Bonn, Kreuzbergweg 26, D-53115 Bonn, Germany
3 Institute of General and Ecological Chemistry, Technical University of Łódz´, Żwirki 36, Pl 30-924 Łódz´, Poland
4 University of Hannover, Institute of Organic Chemistry, Schneiderberg 1B, D-30167 Hannover, Germany

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  • Drabczyńska Anna, Karcz Tadeusz, Szymańska Ewa, Köse Meryem, Müller Christa E., Paskaleva Minka, Karolak-Wojciechowska Janina, Handzlik Jadwiga, Yuzlenko Olga, Kieć-Kononowicz Katarzyna: Synthesis, biological activity and molecular modelling studies of tricyclic alkylimidazo-, pyrimido- and diazepinopurinediones. Purinergic Signalling 2013, 9, 395. <http://dx.doi.org/10.1007/s11302-013-9358-3>
  • Drabczyńska Anna, Yuzlenko Olga, Köse Meryem, Paskaleva Minka, Schiedel Anke C., Karolak-Wojciechowska Janina, Handzlik Jadwiga, Karcz Tadeusz, Kuder Kamil, Müller Christa E.: Synthesis and biological activity of tricyclic cycloalkylimidazo-, pyrimido- and diazepinopurinediones. Eur Med Chem 2011, 46, 3590. <http://dx.doi.org/10.1016/j.ejmech.2011.05.023>
  • Kawczak Piotr, Vander Heyden Yvan, Nasal Antoni, Bączek Tomasz, Drabczyñska Anna, Kieć-Kononowicz Katarzyna, Kaliszan Roman: Micellar liquid chromatography for lipophilicity determination of new biologically active 1,3-purinodiones. J Sep Science 2010, 33, 1546. <http://dx.doi.org/10.1002/jssc.200900752>
  • Ye Deju, Zhang Xu, Zhou Yu, Zhang Dengyou, Zhang Lei, Wang Hengshuai, Jiang Hualiang, Liu Hong: Gold- and Silver-Catalyzed Intramolecular Hydroamination of Terminal Alkynes: Water-Triggered Chemo- and Regioselective Synthesis of Fused Tricyclic Xanthines. Adv Synth Catal 2009, 351, 2770. <http://dx.doi.org/10.1002/adsc.200900505>
  • Yuzlenko Olga, Kieć-Kononowicz Katarzyna: Molecular modeling of A1 and A2A adenosine receptors: Comparison of rhodopsin- and β2-adrenergic-based homology models through the docking studies. J Comput Chem 2009, 30, 14. <http://dx.doi.org/10.1002/jcc.21001>
  • Yuzlenko Olga, Drabczyńska Anna, Kieć-Kononowicz Katarzyna: Predictive 3D-Quantitative Structure-Activity Relationship for A1 and A2A Adenosine Receptor Ligands. QSAR Comb Sci 2009, 28, 1442. <http://dx.doi.org/10.1002/qsar.200910047>
  • González Maykel Pérez, Terán Carmen, Teijeira Marta: Search for new antagonist ligands for adenosine receptors from QSAR point of view. How close are we?. Med Res Rev 2008, 28, 329. <http://dx.doi.org/10.1002/med.20108>
  • González Maykel Pérez, Terán Carmen, Teijeira Marta, Helguera Aliuska Morales: QSAR Studies Using Radial Distribution Function for Predicting A1 Adenosine Receptors Agonists. Bull Math Biol 2007, 69, 347. <http://dx.doi.org/10.1007/s11538-006-9127-3>
  • Drabczyńska Anna, Müller Christa E., Karolak-Wojciechowska Janina, Schumacher Britta, Schiedel Anke, Yuzlenko Olga, Kieć-Kononowicz Katarzyna: N9-Benzyl-substituted 1,3-dimethyl- and 1,3-dipropyl-pyrimido[2,1-f]purinediones: Synthesis and structure–activity relationships at adenosine A1 and A2A receptors. biorg med chem 2007, 15, 5003. <http://dx.doi.org/10.1016/j.bmc.2007.04.018>
  • Drabczyńska Anna, Müller Christa E., Schiedel Anke, Schumacher Britta, Karolak-Wojciechowska Janina, Fruziński Andrzej, Zobnina Weronika, Yuzlenko Olga, Kieć-Kononowicz Katarzyna: Phenylethyl-substituted pyrimido[2,1-f]purinediones and related compounds: Structure–activity relationships as adenosine A1 and A2A receptor ligands. biorg med chem 2007, 15, 6956. <http://dx.doi.org/10.1016/j.bmc.2007.07.051>
  • Drabczyńska Anna, Müller Christa E., Lacher Svenja K., Schumacher Britta, Karolak-Wojciechowska Janina, Nasal Antony, Kawczak Piotr, Yuzlenko Olga, Pękala Elżbieta, Kieć-Kononowicz Katarzyna: Synthesis and biological activity of tricyclic aryloimidazo-, pyrimido-, and diazepinopurinediones. Bioorganic & Medicinal Chemistry 2006, 14, 7258. <http://dx.doi.org/10.1016/j.bmc.2006.06.052>
  • Chabchoub Fakher, Rekik Awatef, Salem Mansour: Heterocyclization of Imidates with 3‐Alkyl‐5‐amino‐1‐phenyl‐1,2,4‐triazoles: Synthesis of New Triazolotriazines. Synth Common 2005, 35, 2467. <http://dx.doi.org/10.1080/00397910500191334>
  • Drabczyńska Anna, Müller Christa E., Schumacher Britta, Hinz Sonja, Karolak-Wojciechowska Janina, Michalak Barbara, Pękala Elżbieta, Kieć-Kononowicz Katarzyna: Tricyclic oxazolo[2,3-f]purinediones: potency as adenosine receptor ligands and anticonvulsants. biorg med chem 2004, 12, 4895. <http://dx.doi.org/10.1016/j.bmc.2004.06.043>
  • Schumacher Britta, Müller Christa E., Karolak-Wojciechowska Janina, Michalak Barbara, Pękala Elżbieta, Kieć-Kononowicz Katarzyna, Drabczyńska Anna: Impact of the aryl substituent kind and distance from pyrimido[2,1-f]purindiones on the adenosine receptor selectivity and antagonistic properties. Eur J Med Chem 2003, 38, 397. <http://dx.doi.org/10.1016/S0223-5234(03)00051-5>