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Pure Appl. Chem., 1996, Vol. 68, No. 6, pp. 1303-1308

Peptidomimetic building blocks for drug discovery: An overview

M. Goodman and H. Shao

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  • Shirakawa Seiji, Liu Yan, Usui Asuka, Maruoka Keiji: Efficient Asymmetric Synthesis of a Bicyclic Amino Acid as a Core Structure of Telaprevir. ChemCatChem 2012, 4, 980. <>
  • Moro Stefano, Floris Matteo: Mimicking Peptides… In Silico. Mol Inf 2012, 31, 12. <>
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  • Sridevi C., Panneer Selvam N., Shanthi G., Velraj G.: Tautomeric stability, vibrational, electronic, NBO, and NMR analyses of N-[acetylamino-(3-nitrophenyl)methyl]-acetamide (ANPMA) by ab initio HF and DFT calculations. Journal of Molecular Structure 2012, 1030, 46. <>
  • Mohite Amar R., Bhat Ramakrishna G.: Enantiopure Synthesis of Side Chain-Modified α-Amino Acids and 5-cis-Alkylprolines. J. Org. Chem. 2012, 77, 5423. <>
  • Terrasson Vincent, Campagne Jean Marc, Moreau Xavier, Greck Christine, Marcia de Figueiredo Renata, Desmarchelier Alaric, Pereira de Sant'Ana Danilo: Organocatalyzed Aziridination of α-Branched Enals: Enantioselective Synthesis of Aziridines with a Quaternary Stereo­center. Eur J Org Chem 2011, 2011, 4046. <>
  • Kuriata-Adamusiak Renata, Strub Daniel, Szatkowski Paweł, Lochyński Stanisław: Biotransformation of bicyclic terpenoid ketones towards compounds with olfactory properties : Biotransformation of bicyclic terpenoid ketones. Flavour Fragr J 2011, n/a. <>
  • GOODMAN M., SHAO H.: ChemInform Abstract: Peptidomimetic Building Blocks for Drug Discovery: An Overview. ChemInform 2010, 28, no. <>
  • Sundararaju Basker, Sridhar Tailor, Achard Mathieu, Sharma Gangavaram V. M., Bruneau Christian: Preparation of Sugar β-Amino Acid Derivatives with Cyclic Structures by Ring-Closing Metathesis. Eur J Org Chem 2010, 2010, 6092. <>
  • Ranatunga Sujeewa, Valle Juan R. Del: Synthesis of Boc-protected bicycloproline. Tetrahetron Lett 2009, 50, 2464. <>
  • MAYER JOHN P., ZHANG JINGWEN, GROEGER STEFAN, LIU CHUAN-FA, JAROSINSKI MARK A.: Lanthionine macrocyclization by in situ activation of serine. J Pept Res 2009, 51, 432. <>
  • Undheim K.: The Schöllkopf chiron and transition metal mediated reactions, a powerful combination for stereoselective construction of cyclic α-quaternary-α-amino acid derivatives. Amino Acids 2008, 34, 357. <>
  • Aydillo Carlos, Avenoza Alberto, Busto Jesús H., Jiménez-Osés Gonzalo, Peregrina Jesús M., Zurbano María M.: α-Alkylation versus retro-O-Michael/γ-alkylation of bicyclic N,O-acetals: an entry to α-methylthreonine. Tet Asymm 2008, 19, 2829. <>
  • Nugent Thomas C., Ghosh Abhijit K.: Selective Synthesis of Unnatural α-, β- and γ-Amino Esters. Eur J Org Chem 2007, 2007, 3863. <>
  • Andrei Mioara, Efskind Jon, Undheim Kjell: A stereoselective synthesis of a spiro-bridged bis(α-amino acid) derivative based on Ru(II)-catalysed RCM reactions. Tetrahedron 2007, 63, 4347. <>
  • Toniolo Claudio: From coded to non-coded α-amino acids: a journey in oligopeptide stereochemistry. J Peptide Sci 2005, 11, 250. <>
  • Furenes Eline Bredal, Luijendijk Jaco, Efskind Jon, Undheim Kjell: Synthesis of Benzene‐1‐Alanine‐3‐Glycine as Carba Analogues of Cystine. Synth Common 2005, 35, 193. <>
  • Qiu Xiao-Long, Meng Wei-Dong, Qing Feng-Ling: Synthesis of fluorinated amino acids. Tetrahedron 2004, 60, 6711. <>
  • Avenoza Alberto, Busto Jesús H., Corzana Francisco, Peregrina Jesús M., Sucunza David, Zurbano Marı́a M.: α-Methylserinals as an access to α-methyl-β-hydroxyamino acids: application in the synthesis of all stereoisomers of α-methylthreonine. Tet Asymm 2004, 15, 719. <>
  • Andrei Mioara, Efskind Jon, Viljugrein Trine, Rømming Christian, Undheim Kjell: Chemoselective rhodium(II)–carbenoid cyclisation reactions in the stereoselective construction of rigidified cyclic α-amino acid derivatives. Tet Asymm 2004, 15, 1301. <>
  • Matteucci Mizio, Bhalay Gurdip, Bradley Mark: Cystine mimetics––solid phase lanthionine synthesis. Tetrahetron Lett 2004, 45, 1399. <>
  • Cetina M., Dzolic Z., Mrvos-Sermek D., Hergold-Brundic A., Nagl A., Mintas M.: Synthesis and X-ray study of the 6-(N-pyrrolyl)purine and thymine derivatives of 1-aminocyclopropane-1-carboxylic acid. J Pept Res 2004, 63, 391. <>
  • Schumacher Marc, Miesch Laurence, Franck-Neumann Michel: Diene(tricarbonyl)iron complexes linked to spirooxazolones for the synthesis of cyclopropyldihydroxyphenylalanine. Tetrahetron Lett 2003, 44, 5393. <>
  • Møller Bjørg S., Undheim Kjell: A Versatile Method for the Preparation of Enantiomeric Benzene-1,2-bis(alanine) Derivatives. Synth Common 2003, 33, 4209. <>
  • Park Kyung-Ho, Kurth Mark J.: Cyclic amino acid derivatives. Tetrahedron 2002, 58, 8629. <>
  • Krikstolaityté Sonata, Hammer Kristin, Rømming Christian, Undheim Kjell: SYNTHESIS OF CYCLIC CONSTRAINED β-OXO-SUBSTITUTED α-AMINO ACIDS. Synth Common 2002, 32, 571. <>
  • Goodman Murray, Zapf Christoph, Rew Yosup: New reagents, reactions, and peptidomimetics for drug design. Biopolymers (Biospectroscopy) 2001, 60, 229. <<229::AID-BIP10034>3.0.CO;2-P>
  • Lane Jonathan W, Halcomb Randall L: New design concepts for constraining glycosylated amino acids. Tetrahedron 2001, 57, 6531. <>
  • Kotha Sambasivarao, Sreenivasachary Nampally, Brahmachary Enugurthi: Synthesis of benzocycloheptene-based amino acid derivatives via a [4+2] cycloaddition reaction as a key step. Tetrahedron 2001, 57, 6261. <>
  • Vera-Ayoso Yolanda, Borrachero Pastora, Cabrera-Escribano Francisca, Diánez Ma̱ Jesús, Estrada Ma̱ Dolores, Gómez-Guillén Manuel, López-Castro Amparo, Pérez-Garrido Simeón: Towards cyclic, conformationally constrained, fluorine-containing β-amino acid derivatives from d-glucose. Tet Asymm 2001, 12, 2031. <>
  • Kotha Sambasivarao, Sreenivasachary Nampally, Mohanraja Kumar, Durani Susheel: Modification of constrained peptides by ring-closing metathesis reaction. Biorg Med Chem Lett 2001, 11, 1421. <>
  • OHWADA Tomohiko: Nitrogen Pyramidal Amides and Related Compounds. YAKUGAKU ZASSHI 2001, 121, 65. <>
  • Undheim Kjell: Stereoselective routes towards the synthesis of unusual bis(amino acids) and cyclic amino acids. Lett Peptide Sci 1998, 5, 227. <>
  • Lange Meinolf, Undheim Kjell: Stereoselective synthesis of α,α′-bridged bis(α-alanine) derivatives. Tetrahedron 1998, 54, 5337. <>
  • Lange Meinolf, Pettersen Anne Lise, Undheim Kjell: Synthesis of secondary amines by reductive dimerization of azides. Tetrahedron 1998, 54, 5745. <>
  • Ohwada Tomohiko, Achiwa Takuji, Okamoto Iwao, Shudo Koichi, Yamaguchi Kentaro: On the planarity of amide nitrogen. Intrinsic pyramidal nitrogen of N-acyl-7-azabicyclo[2.2.1]heptanes. Tetrahetron Lett 1998, 39, 865. <>
  • Krikstolaitytè Sonata, Hammer Kristin, Undheim Kjell: Ru(II)-catalyzed RCM reactions with electrophilic diene substrates. Tetrahetron Lett 1998, 39, 7595. <>
  • Goodman Murray, Zhang Jinfang, Gantzel Peter, Benedetti Ettore: The stereocontrolled synthesis of orthogonally protected (R)-α-methyltryptophan. Tetrahetron Lett 1998, 39, 9589. <>
  • Hammer Kristin, Undheim Kjell: Ruthenium(II) in ring closing metathesis for the stereoselective preparation of cyclic 1-amino-1-carboxylic acids. Tetrahedron 1997, 53, 2309. <>
  • Hammer Kristin, Undheim Kjell: Synthesis of conformationally restricted serine derivatives through ruthenium(II)-catalyzed ring closing metathesis. Tetrahedron 1997, 53, 5925. <>
  • Neset Siren, Hope Håkon, Undheim Kjell: Stereoselective synthesis of cyclopropane-1,2-bis(glycine) derivatives. Tetrahedron 1997, 53, 10459. <>
  • Hammer Kristin, Undheim Kjell: Ruthenium-catalyzed enyne metathesis in stereoselective preparation of cyclic 1-amino-1-carboxylic acids. Tetrahedron 1997, 53, 10603. <>